57801-95-3
Product Description
https://www.krt-chemical.com/products/flubrotizolam-cas-57801-95-3.html
Fluorobrotizolam is a synthetic benzodiazepine and thienodiazepine derivative that has recently emerged as a new psychoactive substance. It is a potent hypnotic with sedative, anxiolytic, anticonvulsant and muscle relaxant effects. Flubromtizolam is structurally related to other benzodiazepines (e.g., flubromazolam, diazepam, and clonazolam) and is thought to have a similar pharmacological profile. This paper will provide an overview of the synthetic methodology, scientific research applications, mechanism of action, biochemical and physiological effects, advantages and limitations of laboratory experiments, and future directions of flurbromotizolam.
Scientific Research Applications
Flubendazolam has been studied for use in scientific research. Flubendazolam has been found to be effective in the treatment of anxiety and insomnia, as well as a potential treatment for a variety of neurological disorders. It has also been studied for the treatment of pain, epilepsy, and addiction. In addition, Flubendazolam has been studied for the treatment of depression, bipolar disorder and schizophrenia.
Mechanism of action
Flurbotizolam is thought to be an orthosteric modulator of GABA-A receptors, the major inhibitory neurotransmitter in the central nervous system. This effect of flurbutizolam is thought to be responsible for its anxiolytic, hypnotic, anticonvulsant, and muscle relaxant effects. In addition, flurbutizolam is thought to be an inverse agonist at the 5-HT2A receptor, the main excitatory neurotransmitter in the central nervous system. This effect of flurbutizolam is thought to be responsible for its sedative effects.
Biochemical and Physiological Effects
Flurbutizolam has been found to produce a variety of biochemical and physiological effects. It has been found to increase the activity of GABA-A receptors, which enhances CNS depression. This effect of flurbutizolam is responsible for its anxiolytic, hypnotic, anticonvulsant and muscle relaxant effects. In addition, Flurbutizolam has been found to decrease the activity of 5-HT2A receptors, which results in decreased excitability of the central nervous system. This effect of flurbutizolam is responsible for its sedative effects.
Flubrotizolam is a thienotriazolodiazepine derivative with potent sedative and anxiolytic effects, which has been sold as a designer drug.
Formal Name
2-bromo-4-(2-fluorophenyl)-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine
CAS Number 57801-95-3
Molecular Formula C15H10BrFN4S
Formula Weight 377.2
Purity ≥98%
Formulation (Request formulation change) A crystalline solid
Solubility (Learn about Variance in Solubility)DMF: 5 mg/ml DMSO: 5 mg/ml DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml
Λmax 244 nm
SMILES CC1=NN=C2CN=C(C3=CC=CC=C3F)C4=C(SC(Br)=C4)N21
Shipping & Storage Information
Storage -20°C
Shipping Room Temperature in continental US; may vary elsewhere
Stability ≥ 2 years
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